Product Name: A-286501
Description: A-286501 is a novel orally active adenosine kinase inhibitor (IC50=0.47 nM). A-286501 was orally effective to reduce nociception in animal models of acute (thermal), inflammatory (formalin and carrageenan), and neuropathic (L5/L6 nerve ligation and strep
CAS NO: 516-54-1 Product: Allopregnanolone
Synonym: A-286501; A 286501; A286501.
IUPAC Chemical Name: (1S,2R,3S,5R)-3-amino-5-(4-amino-5-bromo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)cyclopentane-1,2-diol
In ChiKey: FKFYQPGMXTXSTC-LWIVVEGESA-NEpigenetics inhibitors
SMILE Code: BrC(C1=C2N=CN=C1N)=CN2[C@H]3[C@H](O)[C@H](O)[C@@H](N)C3
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Web Site click
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22110104
Chemical Formula:C11H14BrN5O2
ExactMass: 327.0331
Molecular Weight: 328.17
Elemental Analysis: C, 40.26; H, 4.30; Br, 24.35; N, 21.34; O, 9.75
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