Product Name: E-52862 HCl featured
Description: E-52862, also known as S1RA, is a selective sigma-1 receptor antagonist, with a reported binding affinity of Ki = 17.0 ± 7.0 nM, selective over the sigma-2 receptor and against a panel of other 170 receptors, enzymes, transporters and ion channels. In p
CAS NO: 1448440-52-5 Product: SP-13786
Synonym: E-52862; E 52862; E52862; S1RA; E-52862 HCl; E-52862 hydrochloride; S1RA hydrochloride.
IUPAC Chemical Name: 4-(2-((5-methyl-1-(naphthalen-2-yl)-1H-pyrazol-3-yl)oxy)ethyl)morpholine hydrochloride
In ChiKey: SHRYQZBTQDMGLZ-UHFFFAOYSA-NItk inhibitors
SMILE Code: CC1=CC(OCCN2CCOCC2)=NN1C3=CC=C4C=CC=CC4=C3.[H]Cl
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Web Site：Medchemexpress
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22118073
Chemical Formula：C20H24ClN3O2
ExactMass: 337.179
Molecular Weight: 373.881
Elemental Analysis: C, 64.25; H, 6.47; Cl, 9.48; N, 11.24; O, 8.56
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