Product Name: Farglitazar
Description: Farglitazar, also known as GI-262570, is a PPAR-γ agonist potentially for the treatment of type 2 diabetes. GI262570 can increase water and sodium reabsorption in distal nephron by stimulating the ENaC and Na,K-ATPase system.
CAS NO: 1198786-98-9 Product: INT-777 (R-enantiomer)
Synonym: Farglitazar; GI-262570; GI 262570; GI262570.
IUPAC Chemical Name: (S)-2-((2-benzoylphenyl)amino)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)propanoic acid
In ChiKey: Cell_Counting_Kit-8 inhibitors
SMILE Code: O=C(O)[C@H](CC1=CC=C(OCCC2=C(C)OC(C3=CC=CC=C3)=N2)C=C1)NC4=CC=CC=C4C(C5=CC=CC=C5)=O
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress.com
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22120009
Chemical Formula：C34H30N2O5
ExactMass: 546.2155
Molecular Weight: 546.623
Elemental Analysis: C, 74.71; H, 5.53; N, 5.12; O, 14.63
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