Product Name: Galeterone new featured
Description: Galeterone, also known as TOK-001 and NX41765; is an orally bioavailable small-molecule androgen receptor modulator and CYP17 lyase inhibitor with potential antiandrogen activity. Galeterone exhibits three distinct mechanisms of action: 1) as an androgen
CAS NO: 55224-05-0 Product: Erythromycin Cyclocarbonate
Synonym: TOK001; TOK 001; TOK-001; NX41765; NX 41765; NX-41765; VN 1241; VN-1241; VN-1241; Galeterone.
IUPAC Chemical Name: (3S,8R,9S,10R,13S,14S)-17-(1H-benzo[d]imidazol-1-yl)-10,13-dimethyl-2,3,4,7,8,9,10,11,12,13,14,15-dodecahydro-1H-cyclopenta[a]phenanthren-3-ol
In ChiKey: PAFKTGFSEFKSQG-PAASFTFBSA-NCasein Kinase inhibitors
SMILE Code: O[C@H]1CC[C@]2(C)[C@@]3([H])CC[C@]4(C)C(N5C=NC6=CC=CC=C56)=CC[C@@]4([H])[C@]3([H])CC=C2C1
Appearance: White to off white solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22122083
Chemical Formula：C26H32N2O
ExactMass: 388.25146
Molecular Weight: 388.54508
Elemental Analysis: C, 80.37; H, 8.30; N, 7.21; O, 4.12
bet-bromodomain.com
BET Bromodomain Inhibitor
