Product Name: HC-030031
Description: HC-030031 is a potent and selective TRPA1 antagonist, attenuates inflammatory- and neuropathy-induced mechanical hypersensitivity. HC-030031 antagonizes AITC- and formalin-evoked calcium influx with IC50 of 6.2 μM and 5.3 μM respectively.
CAS NO: 863971-12-4 Product: MMAF-OMe
Synonym: HC-030031; HC 030031; HC030031.
IUPAC Chemical Name: 2-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)-N-(4-isopropylphenyl)acetamide
In ChiKey: GHSR inhibitors
SMILE Code: O=C(NC1=CC=C(C(C)C)C=C1)CN2C=NC(N(C)C(N3C)=O)=C2C3=O
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Web Site:Medchemexpress
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22124249
Chemical Formula:C18H21N5O3
ExactMass: 355.1644
Molecular Weight: 355.398
Elemental Analysis: C, 60.83; H, 5.96; N, 19.71; O, 13.51
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