Product Name: JD5037
Description: JD5037 is a peripherally restricted (PR) cannabinoid-1 receptor blocker. JD5037 is an antiobesity drug candidate which acts as a peripherally-restricted cannabinoid inverse agonist at CB1 receptors. It is very selective for the CB1 subtype, with a Ki of
CAS NO: 1642300-52-4 Product: KPT-8602
Synonym: JD5037; JD-5037; JD 5037.
IUPAC Chemical Name: (S)-2-(((E)-((S)-3-(4-chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazol-1-yl)((4-chlorophenyl)sulfonamido)methylene)amino)-3-methylbutanamide
In ChiKey: GTCSIQFTNPTSLO-RPWUZVMVSA-NMetabolic Enzyme_Protease inhibitors
SMILE Code: CC(C)[C@@H](C(N)=O)/N=C(N1N=C(C2=CC=C(Cl)C=C2)[C@@H](C3=CC=CC=C3)C1)/NS(=O)(C4=CC=C(Cl)C=C4)=O
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Web Site click
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22127587
Chemical Formula：C27H27Cl2N5O3S
ExactMass: 571.1212
Molecular Weight: 572.505
Elemental Analysis: C, 56.65; H, 4.75; Cl, 12.38; N, 12.23; O, 8.38; S, 5.60
bet-bromodomain.com
BET Bromodomain Inhibitor
