Product Name: JNJ-17156516
Description: JNJ-17156516 is a novel, potent, and selective cholecystokinin 1 receptor antagonist. JNJ-17156516 expressed high-affinity at the cloned human (pK(I) = 7.96 +/- 0.11), rat (pK(I) = 8.02 +/- 0.11), and canine (pK(I) = 7.98 +/- 0.04) CCK1 receptors, and it
CAS NO: 1008763-54-9 Product: D-3263 (hydrochloride)
Synonym: JNJ-17156516; JNJ 17156516; JNJ17156516.
IUPAC Chemical Name: (S)-3-(5-(3,4-Dichlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-3-yl)-2-(3-methylphenyl)propionic acid
In ChiKey: Farnesyl Transferase inhibitors
SMILE Code: O=C(O)[C@H](C1=CC=CC(C)=C1)CC2=NN(C3=CC=C(OC)C=C3)C(C4=CC=C(Cl)C(Cl)=C4)=C2
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Web Site:Medchemexpress
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22128219
Chemical Formula:C26H22Cl2N2O3
ExactMass: 480.10075
Molecular Weight: 481.37
Elemental Analysis: C, 64.87; H, 4.61; Cl, 14.73; N, 5.82; O, 9.97
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