Product Name: M77976
Description: M77976 is a PDK4 inhibitor (human pyruvate dehydrogenase kinase 4). M77976 binds to the ATP-binding pocket of PDK4 and causes local conformational changes with complete disordering of the ATP lid. M77976 binding also leads to a large domain rearrangement
CAS NO: 97657-92-6 Product: Latrepirdine (dihydrochloride)
Synonym: M77976; M-77976; M 77976.
IUPAC Chemical Name: 4-(4-(4-methoxyphenyl)-5-methyl-1H-pyrazol-3-yl)benzene-1,3-diol
In ChiKey: GSBFARPNIZUMHA-UHFFFAOYSA-NStem_Cell_Signaling_Compound_Library inhibitors
SMILE Code: COC1=CC=C(C2=C(C)NN=C2C3=CC=C(O)C=C3O)C=C1
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress.com
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22133255
Chemical Formula：C17H16N2O3
ExactMass: 296.1161
Molecular Weight: 296.326
Elemental Analysis: C, 68.91; H, 5.44; N, 9.45; O, 16.20
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