Product Name: Macimorelin
Description: Macimorelin, also known as AEZS-130, EP-1572, or JMV1843, is a novel synthetic small molecule, acting as a ghrelin agonist, that is orally active and stimulates the secretion of growth hormone (GH). Based on results of Phase 1 studies, AEZS-130 has poten
CAS NO: 1808011-22-4 Product: EPZ031686
Synonym: JMV1843; JMV-1843; JMV 1843; AEZS-130; AEZS 130; AEZS130; EP-1572; EP 1572; EP1572; UMV-1843; UMV 1843; Macimorelin; AibDTrpDgTrpCHO.
IUPAC Chemical Name: 2-amino-N-((R)-1-(((R)-1-formamido-2-(1H-indol-3-yl)ethyl)amino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)-2-methylpropanamide
In ChiKey: UJVDJAPJQWZRFR-DHIUTWEWSA-NWnt/Hedgehog/Notch_Compound_Library inhibitors
SMILE Code: CC(C)(N)C(N[C@H](CC1=CNC2=C1C=CC=C2)C(N[C@@H](NC=O)CC3=CNC4=C3C=CC=C4)=O)=O
Appearance: white solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22133283
Chemical Formula:C26H30N6O3
ExactMass: 474.23794
Molecular Weight: 474.5548
Elemental Analysis: C, 65.80; H, 6.37; N, 17.71; O, 10.11
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