Product Name: OK-1035
Description: OK-1035 is a potent and selective DNA-PK inhibitor. When a synthetic peptide was used as a substrate, OK-1035 caused 50% inhibition of DNA-PK activity at 8 microM. OK-1035 inhibited the phosphorylation by DNA-PK of consensus peptide as well as that of rec
CAS NO: 1439901-97-9 Product: ONO-4059 (hydrochloride)
Synonym: OK1035; OK 1035; OK-1035.
IUPAC Chemical Name: (E)-2-(hydrazonomethyl)-6-oxo-1,6-dihydro-[3,4-bipyridine]-5-carbonitrile
In ChiKey: GPR119 inhibitors
SMILE Code: N#CC1=CC(C2=CC=NC=C2)=C(/C=N/N)NC1=O
Appearance: white solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress.com
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22138161
Chemical Formula:C12H9N5O
ExactMass: 239.08071
Molecular Weight: 239.23276
Elemental Analysis: C, 60.25; H, 3.79; N, 29.27; O, 6.69
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