Product Name: S-8510 free base
Description: S-8510, also known as SB-737552, is a GABA-A receptor inverse agonist potentially for the treatment of dementia. S-8510 ameliorated memory impairment induced by cholinergic deficit in the water maze paradigm of Wistar rats. S-8510 augmented LTP of the Sch
CAS NO: 415903-37-6 Product: Grapiprant
Synonym: S-8510; SB-737552; S8510; SB737552; S 8510; SB 737552.
IUPAC Chemical Name: 2-(isoxazol-3-yl)-1,6,7,9-tetrahydroimidazo[4,5-d]pyrano[4,3-b]pyridine
In ChiKey: RGS Protein inhibitors
SMILE Code: C12=NC=C3C(NC(C4=NOC=C4)=N3)=C1COCC2
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Web Site click
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22145475
Chemical Formula:C12H10N4O2
ExactMass: 242.0804
Molecular Weight: 242.238
Elemental Analysis: C, 59.50; H, 4.16; N, 23.13; O, 13.21
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