Product Name: Sacubitrilat featured
Description: Sacubitrilat, also known as LBQ-657, is endopeptidase inhibitor. Sacubitril is a prodrug that is activated to LBQ657 by de-ethylation via esterases. LBQ657 inhibits the enzyme neprilysin, which is responsible for the degradation of atrial and brain natri
CAS NO: 1174018-99-5 Product: Relebactam
Synonym: LBQ-657; LBQ 657; LBQ657; Sacubitrilat.
IUPAC Chemical Name: (2R,4S)-5-([1,1-biphenyl]-4-yl)-4-(3-carboxypropanamido)-2-methylpentanoic acid
In ChiKey: DOBNVUFHFMVMDB-BEFAXECRSA-NImmunology_Inflammation inhibitors
SMILE Code: O=C(O)[C@H](C)C[C@H](NC(CCC(O)=O)=O)CC1=CC=C(C2=CC=CC=C2)C=C1
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress.com
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22145804
Chemical Formula：C22H25NO5
ExactMass: 383.1733
Molecular Weight: 383.444
Elemental Analysis: C, 68.91; H, 6.57; N, 3.65; O, 20.86
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