Product Name: T-98475
Description: T-98475 is a potent, orally active and non-peptide gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist (IC50 values are 0.2, 4.0 and 60 nM for human, monkey and rat GnRH receptors respectively). T-98475 inhibits LH release in vitro (IC50 = 100
CAS NO: 1627709-94-7 Product: LJI308
Synonym: T-98475; T 98475; T98475.
IUPAC Chemical Name: propan-2-yl 7-[(2,6-difluorophenyl)methyl]-3-[(methyl-(phenylmethyl)amino)methyl]-2-[4-(2-methylpropanoylamino)phenyl]-4-oxothieno[3,2-e]pyridine-5-carboxylate
In ChiKey: RANJJVIMTOIWIN-UHFFFAOYSA-NMonoamine Transporter inhibitors
SMILE Code: O=C(C1=CN(CC2=C(F)C=CC=C2F)C3=C(C(CN(C)CC4=CC=CC=C4)=C(C5=CC=C(NC(C(C)C)=O)C=C5)S3)C1=O)OC(C)C
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Web Site click
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22147520
Chemical Formula：C37H37F2N3O4S
ExactMass: 657.2473
Molecular Weight: 657.78
Elemental Analysis: C, 67.56; H, 5.67; F, 5.78; N, 6.39; O, 9.73; S, 4.87
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