Product Name: T0070907 featured
Description: T0070907 was identified as a potent and selective PPARgamma antagonist. With an apparent binding affinity (concentration at 50% inhibition of [(3)H]rosiglitazone binding or IC(50)) of 1 nm, T0070907 covalently modifies PPARgamma on cysteine 313 in helix 3
CAS NO: 1142090-23-0 Product: GSK2256294A
Synonym: T0070907; T-0070907; T 0070907.
IUPAC Chemical Name: 2-chloro-5-nitro-N-(pyridin-4-yl)benzamide
In ChiKey: FRPJSHKMZHWJBE-UHFFFAOYSA-NKLF inhibitors
SMILE Code: O=C(NC1=CC=NC=C1)C2=CC([N+]([O-])=O)=CC=C2Cl
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Web Site:Medchemexpress
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 5 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/221468
Chemical Formula:C12H8ClN3O3
ExactMass: 277.02542
Molecular Weight: 277.66
Elemental Analysis: C, 51.91; H, 2.90; Cl, 12.77; N, 15.13; O, 17.29
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