Product Name: Varespladib (LY315920) featured
Description: Varespladib, aslo known as LY315920, is a secreted phospholipase A2 (sPLA2) inhibitor (IC50 = 50 – 750 nM for a range of sPLA2 isoforms). Varespladib reduces atherosclerosis and aneurysm formation in ApoE-/- mice and in guinea pigs. Varespladib signific
CAS NO: 1532533-78-0 Product: TGR-1202 (hydrochloride)
Synonym: LY315920; LY-315920; LY 315920; A-002; A002; A 002; Varespladib
IUPAC Chemical Name: 2-((3-(2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-indol-4-yl)oxy)acetic acid
In ChiKey: BHLXTPHDSZUFHR-UHFFFAOYSA-NBombesin Receptor inhibitors
SMILE Code: NC(C(C1=C(CC)N(CC2=CC=CC=C2)C3=C1C(OCC(O)=O)=CC=C3)=O)=O
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22152680
Chemical Formula：C21H20N2O5
ExactMass: 380.13722
Molecular Weight: 380.4
Elemental Analysis: C, 66.31; H, 5.30; N, 7.36; O, 21.03
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