Product Name: Varespladib Methyl
Description: Varespladib Methyl, also known as A-002; LY-333013; S-3013, is a secretory phospholipase A2 (sPLA2) inhibitor as a potential treatment for acute coronary syndrome (ACS). Varespladib methyl is an orally bioavailable prodrug of the molecule varespladib. Va
CAS NO: 1532533-67-7 Product: TGR-1202
Synonym: A-002; A002; A002; LY-333013; LY 333013; LY333013; S-3013; S 3013; S3013; Varespladib Methyl.
IUPAC Chemical Name: methyl 2-((3-(2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-indol-4-yl)oxy)acetate
In ChiKey: VJYDOJXJUCJUHL-UHFFFAOYSA-NBradykinin Receptor inhibitors
SMILE Code: O=C(OC)COC1=CC=CC2=C1C(C(C(N)=O)=O)=C(CC)N2CC3=CC=CC=C3
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress.com
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22152767
Chemical Formula:C22H22N2O5
ExactMass: 394.1529
Molecular Weight: 394.427
Elemental Analysis: C, 66.99; H, 5.62; N, 7.10; O, 20.28
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