Product Name: XMD8-87 new featured
Description: XMD8-87 is a TNK2 inhibitor. XMD8-87 showed activity in the inhibition of TNK2 phosphorylation. XMD8-87 and XMD16-5 potently inhibit phosphorylation of TNK2 truncation mutations found in solid tumor types.
CAS NO: 140898-91-5 Product: Hexaminolevulinate (hydrochloride)
Synonym: XMD8-87; XMD-8-87; XMD 8-87; XMD887; XMD-887; XMD 887. ACK1-B19
IUPAC Chemical Name: 2-((2-methoxy-4-(4-methylpiperazin-1-yl)phenyl)amino)-11-methyl-5,11-dihydro-6H-benzo[e]pyrimido[5,4-b][1,4]diazepin-6-one
In ChiKey: LGLHCXISMKHLIK-UHFFFAOYSA-NOrexin Receptor OX Receptor) inhibitors
SMILE Code: C1=NC(NC2=CC=C(N3CCN(C)CC3)C=C2OC)=NC2N(C)C3C=CC=CC=3C(=O)NC1=2
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress.com
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22154369
Chemical Formula：C24H27N7O2
ExactMass: 445.2226
Molecular Weight: 445.527
Elemental Analysis: C, 64.70; H, 6.11; N, 22.01; O, 7.18
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