Product Name: A-770041 featured
Description: A-770041 is a potent ans selective LCK inhibitor. Concanavalin A-stimulated IL-2 production in whole blood is inhibited by A-770041 with an EC50 of approximately 80 nM. A-770041 is orally bioavailable (F = 34.1 +/- 7.2% at 10 mg/kg) and has a t(1/2) of 4
CAS NO: 77472-98-1 Product: Pipequaline
Synonym: A-770041; A 770041; A770041.
IUPAC Chemical Name: (Z)-N-(4-(1-((1r,4r)-4-(4-acetylpiperazin-1-yl)cyclohexyl)-4-amino-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-1-methyl-1H-indole-2-carbimidic acid
In ChiKey: ZMNWFTYYYCSSTF-SOAUALDESA-NEBI2_GPR183 inhibitors
SMILE Code: O/C(C(N1C)=CC2=C1C=CC=C2)=NC3=CC=C(C4=NN([C@H]5CC[C@H](N6CCN(C(C)=O)CC6)CC5)C7=NC=NC(N)=C74)C=C3OC
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Web Site：Medchemexpress
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22110694
Chemical Formula：C34H39N9O3
ExactMass: 621.3176
Molecular Weight: 621.746
Elemental Analysis: C, 65.68; H, 6.32; N, 20.28; O, 7.72
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