Product Name: A-867744 featured
Description: A-867744 is a type II PAM with good potency and selectivity. A-867744 showed acceptable pharmacokinetic profile across species and brain levels sufficient to modulate alpha7 nAChRs. In a rodent model of sensory gating, A-867744 normalized gating deficit
CAS NO: 413611-93-5 Product: 10074-G5
Synonym: A-867744; A 867744; A867744.
IUPAC Chemical Name: 4-(5-(4-Chlorophenyl)-2-methyl-3-propionylpyrrol-1-yl)benzenesulfonamide
In ChiKey: ABACVOXFUHDKNZ-UHFFFAOYSA-NLeukotriene Receptor inhibitors
SMILE Code: O=S(C1=CC=C(N2C(C)=C(C(CC)=O)C=C2C3=CC=C(Cl)C=C3)C=C1)(N)=O
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Web Site click
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22111578
Chemical Formula：C20H19ClN2O3S
ExactMass: 402.0805
Molecular Weight: 402.893
Elemental Analysis: C, 59.62; H, 4.75; Cl, 8.80; N, 6.95; O, 11.91; S, 7.96
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