Product Name: Dagrocorat
Description: Dagrocorat, also known as PF-00251802, is a glucocorticoid receptor agonist and potential useful for anti-inflammatory diseases.
CAS NO: Product: MELK-8a (hydrochloride)
Synonym: PF-00251802; PF 00251802; PF00251802; PF-251802; PF 251802; PF251802; Dagrocorat.
IUPAC Chemical Name: (4bR,7S,8aR)-4b-benzyl-7-hydroxy-N-(2-methylpyridin-3-yl)-7-(trifluoromethyl)-4b,5,6,7,8,8a,9,10-octahydrophenanthrene-2-carboxamide
In ChiKey: Xanthine Oxidase inhibitors
SMILE Code: FC([C@]1(O)CC[C@]2(CC3=CC=CC=C3)C4=CC=C(C(NC5=CC=CN=C5C)=O)C=C4CC[C@]2([H])C1)(F)F
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22116695
Chemical Formula:C29H29F3N2O2
ExactMass: 494.2181
Molecular Weight: 494.5582
Elemental Analysis: C, 70.43; H, 5.91; F, 11.52; N, 5.66; O, 6.47
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