Product Name: Edonentan
Description: Edonentan, also known as BMS-207940, is a highly potent and orally active ET(A) selective antagonist. Edonentan is an extremely potent (ET(A) K(i) = 10 pM) and selective (80,000-fold for ET(A) vs ET(B)) antagonist. It is also 150-fold more potent and >
CAS NO: 1640282-31-0 Product: I-CBP112
Synonym: BMS-207940; BMS207940; BMS 207940; Edonentan
IUPAC Chemical Name: N-((2-(((4,5-Dimethyl-3-isoxazolyl)amino)sulfonyl)-4-(2-oxazolyl)(1,1-biphenyl)-2-yl)methyl)-N,3,3-trimethylbutanamide
In ChiKey: Anti-infection_Compound_Library inhibitors
SMILE Code: CC(C)(C)CC(N(CC1=CC(C2=NC=CO2)=CC=C1C3=CC=CC=C3S(=O)(NC4=NOC(C)=C4C)=O)C)=O
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO, not in water
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22119331
Chemical Formula：C28H32N4O5S
ExactMass: 536.2093
Molecular Weight: 536.647
Elemental Analysis: C, 62.67; H, 6.01; N, 10.44; O, 14.91; S, 5.97
bet-bromodomain.com
BET Bromodomain Inhibitor
