Product Name: Ralimetinib mesylate
Description: Ralimetinib, also known as LY2228820, is a potent and selective, ATP-competitive inhibitor of the α- and β-isoforms of p38 MAPK in vitro (IC(50) = 5.3 and 3.2 nmol/L, respectively). In cell-based assays, LY2228820 potently and selectively inhibited phosph
CAS NO: 148554-65-8 Product: Seco Rapamycin (sodium salt)
Synonym: Ralimetinib mesylate; LY2228820; LY-2228820; LY 2228820; LY2228820 dimesylate.
IUPAC Chemical Name: 5-(2-(tert-butyl)-4-(4-fluorophenyl)-1H-imidazol-5-yl)-3-neopentyl-3H-imidazo[4,5-b]pyridin-2-amine dimethanesulfonate
In ChiKey: Adiponectin Receptor inhibitors
SMILE Code: NC1=NC2=CC=C(C3=C(C4=CC=C(F)C=C4)N=C(C(C)(C)C)N3)N=C2N1CC(C)(C)C.CS(=O)(O)=O.CS(=O)(O)=O
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Web Site click
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22143757
Chemical Formula：C26H37FN6O6S2
ExactMass:
Molecular Weight: 612.7364
Elemental Analysis: C, 50.97; H, 6.09; F, 3.10; N, 13.72; O, 15.67; S, 10.46
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