Product Name: Tafetinib
Description: Tafetinib is a vascular endothelial growth factor receptor (VEGFR) inhibitor for the treatment of solid tumors. Tafeinib is also a multi-targeted receptor tyrosine kinase (RTK) inhibitor.
CAS NO: 1798871-31-4 Product: Centrinone-B
Synonym: Tafetinib; SIM-010603; SIM010603; SIM 010603
IUPAC Chemical Name: (Z)-N-(2-(diethylamino)ethyl)-7-(5-fluoro-2-oxoindolin-3-ylidene)-2-methyl-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
In ChiKey: KGSRYTUWXUESJK-FXBPSFAMSA-NVDAC inhibitors
SMILE Code: CCN(CCNC(C1=C(NC2=C1CCC/C2=C3C(NC4=CC=C(C=C/34)F)=O)C)=O)CC
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress.com
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22147841
Chemical Formula:C24H29FN4O2
ExactMass: 424.2275
Molecular Weight: 424.5204
Elemental Analysis: C, 67.90; H, 6.89; F, 4.48; N, 13.20; O, 7.54
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