Product Name: XEN907
Description: XEN907 is a novel spirooxindole NaV1.7 blocker with IC50 of 3 nM. It shows a further 10-fold increase in potency, which represents a promising structure for further optimization efforts in vitro.
CAS NO: 1332295-35-8 Product: Nav1.7-IN-2
Synonym: XEN907; XEN 907; XEN-907.
IUPAC Chemical Name: 1-pentylspiro[6H-furo[2,3-f][1,3]benzodioxole-7,3-indole]-2-one
In ChiKey: PHMRUZIIERITEP-UHFFFAOYSA-NGPR55 inhibitors
SMILE Code: O=C(C12COC3=C1C=C(OCO4)C4=C3)N(CCCCC)C5=C2C=CC=C5
Appearance: Solid powder
Purity: 98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.Medchemexpress.com
Storage Condition: Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: 2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 – 4 C for short term (days to weeks), or -20 C for long term (months).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22153604
Chemical Formula:C21H21NO4
ExactMass: 351.1471
Molecular Weight: 351.4
Elemental Analysis: C, 71.78; H, 6.02; N, 3.99; O, 18.21
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